Notes
Glycogenolysis
Sections
GLYCOGEN
• Body's glucose reserve
• Can be mobilized more quickly/efficiently than fats
• Stored in liver & muscle
• Mobilized during fast (low insulin: glucagon)
ENZYMES OF GLYCOGENOLYSIS
Glycogen phosphorylase
• Breaks alpha (1,4) bonds
Debranching enzyme
• Breaks alpha (1,6) bonds
• Aka alpha 1,6 glucosidase
Glucose 6-phosphatase
• Tissue specific: liver only
GLYCOGENOLYSIS
- Glycogen phosphorylase removes terminal residues of glycogen branches
• Cleaves alpha (1,4) glycosidic bonds until 4 glucose residues remain per branch
• Cleaves 1 glucose residue at a time
• Glycogen + Pi --> Glucose 1-phosphate - Debranching enzymes transfers 3 residues of shortest branches to longer ones
• One glucose residue remains per branch
• Creates more alpha (1,4) linkages for glycogen phosphorylase to hydrolyze - Debranching enzyme cleaves last glucose residue from short branches
• Cleaves alpha (1,6) bond
• Glycogen + H2O --> Glucose
• Releases residue as glucose NOT glucose 1P - Repeat: glycogen phosphorylase & debranching enzyme degrade glycogen to glucose & glucose 1P
LIVER VERSUS MUSCLE: FATES OF GLUCOSE & GLUCOSE 1P
• Both organs: glucose 1P reversibly converts to glucose 6P
Muscle
• Glucose 6P enters glycolysis --> Pyruvate + ATP
• If O2 is present: pyruvate decarboxylation --> acetyl CoA --> aerobic respiration
• If O2 is absent (exercising muscle): anaerobic glycolysis --> lactate
• Both pyruvate fates produce ATP: fuel for muscle cells
• Stores glycogen for its own use
Liver
• Glucose 6-phosphatase: Glucose 6P --> Glucose + Pi (enzyme NOT in muscle)
• Hepatic glucose released into circulation: fuels peripheral tissues (brain & rbc's)
CLINICAL CORRELATION
Von Gierke's Disease (Type I glycogen storage disease)
• Glucose 6-phosphatase deficiency in liver/kidney
• Frequent hypoglycemia: cannot mobilize glycogen during fast
• Treatment: frequent feedings with slowly digested carbohydrates (i.e. uncooked starch) to maintain blood glucose
Full-Length Text
- Here we'll learn how glycogen is mobilized and broken down in the body, and we'll learn the function of glycogen metabolism in two key organs.
- To begin, start a table to learn some key points about glycogen mobilization.
- Denote that glycogen is the body's glucose reserve, and that it can be mobilized more quickly and efficiently than fats.
- Denote that the liver and muscle both store glycogen.
We will distinguish their roles in glycogen degradation shortly.
- Denote that it is mobilized during fasting state when the insulin to glucagon ratio is low.
- Finally, denote that there are three key enzymes involved in glycogen degradation.
- Glycogen phosphorylase, which breaks alpha (1,4) bonds.
- Debranching enzyme, which breaks alpha (1,6) bonds thus it is also known as alpha 1,6-glucosidase.
- Glucose 6-phosphatase, which is a tissue-specific enzyme; later we'll learn how glycogen breakdown is different in liver and muscle.
To begin, let's illustrate glycogen breakdown.
- Draw a branching glycogen polymer bound to glycogenin.
- It comprises glucose residues.
Let's specifically draw the glucose residues of the top branch.
- Label the first four glucose residues.
- Now, draw two terminal glucose residues.
- These terminal residues will be the first to break off.
- Now, label the first four residues of the remaining branches.
- Next, add the terminal glucose-residues to each branch as follows:
- 1 on the second branch,
- 2 on the third branch
- 1 on the last branch.
- This is our starting glycogen substrate.
Now, let's draw the product.
- Redraw our glycogen polymer, but remove the terminal glucose residues in each branch.
- There should be four glucose residues remaining in each branch.
- Now, indicate that the first key enzyme, glycogen phosphorylase, catalyzes this reaction.
- Write that it removes each glucose residue 1 at a time.
- So, in our case, show that this reaction occurs once per glucose residue, for a total of 6 times.
- Show that a phosphate is consumed per glucose residue, each of which is released as glucose 1-phosphate.
- Now, to clarify this point, write that glycogen phosphorylase cleaves alpha (1,4) glycosidic bonds until 4 glucose residues remain in each branch.
How do we cleave these remaining residues?
- Create a small box to show the actions of debranching enzyme.
- Re-draw the ends of the long branches.
- Then, show that debranching enzyme transfers the last 3 residues of the shortest branches to the longer branches.
Let's draw this product.
- Draw our glycogen polymer with two, elongated branches.
- Show that the top branch has the original 4 residues plus the transferred 3 glucose residues.
- Show that the bottom does as well.
- Show that the shortest branches are now only one glucose-residue long.
- Write that debranching enzyme creates more alpha 1,4 linkages, and therefore a more linear chain, for glycogen phosphorylase to hydrolyze.
Now, we'll see how debranching enzyme further debranches the product.
- Establish another insert.
- Draw the branch points of our product.
- Draw the single glucose residues.
- Then, splice them from their branches.
Let's see the final product.
- Redraw glycogen one last time, and remove the last glucose residues of the shorter branches.
- Write that debranching enzyme cleaves these alpha 1,6 bonds.
- Show that it does this one glucose residue at a time, so this reaction occurs 2 times.
- Indicate that one water molecule is consumed per residue, and that each is released as glucose, not glucose 1-phosphate.
- Next, use a series of arrows to show that glycogen phosphorylase and debranching enzyme continue to breakdown glycogen to glucose and glucose 1-phosphate.
Finally, let's learn the fates of glucose and glucose 1-phosphate in the two organs that can synthesize and store glycogen: the liver and muscle.
- First, draw a chart with two columns: liver and muscle.
- Draw glucose 1-phosphate, the product of glycogen phosphorylase, at the top of each column.
- Show that glucose 1-phosphate reversibly converts to glucose 6-phosphate in both organs.
Now, this is where the fates of glycogen products diverge.
Let's start with the muscle.
- Indicate that glucose 6-phosphate enters glycolysis to produce pyruvate and ATP.
- Now, indicate that pyruvate has two fates in the muscle depending on oxygen conditions:
- If oxygen is present, pyruvate decarboxylation produces acetyl CoA, which can then continue through aerobic respiration.
- If oxygen is absent, as in exercising muscle, pyruvate may enter anaerobic glycolysis to produce lactate.
- However, indicate that both of these fates produce energy as ATP.
- To emphasize this point, write that the muscle glycogenolysis produces fuel for muscle cells.
Now, for the liver.
- Indicate that glucose 6-phosphate is dephosphorylated to produce glucose.
- Show that glucose 6-phosphatase catalyzes this reaction, the last key enzyme in glycogen breakdown.
- Now, highlight this enzyme and write that it is NOT in the muscle.
- Next, show that hepatic glucose is released into circulation.
- Why?
- The brain and red blood cells are glucose-requiring tissues.
- They must use glucose for energy and depend on hepatic glycogen when blood glucose is low.
- Finally, write that hepatic glucose fuels peripheral tissues, particularly the brain and red blood cells.
- The muscle, however, stores glycogen for its own use.
- As a clinical correlation, write that Von Gierke's Disease (Type I glycogen storage disease), is a glucose 6-phosphatase deficiency in the liver and kidney.
- Patients experience frequent hypoglycemia because they cannot mobilize glycogen in times of fast.
- The most common treatment involves frequent feedings with carbohydrates that are very slowly digested, such as uncooked cornstarch, so that blood glucose levels remain within a normal range.